Fluorescence High-Throughput Screening for Inhibitors of TonB Action
نویسندگان
چکیده
منابع مشابه
Fluorescence resonance energy transfer assay for high-throughput screening of ADAMTS1 inhibitors.
A disintegrin and metalloprotease with thrombospondin type I motifs-1 (ADAMTS1) plays a crucial role in inflammatory joint diseases and its inhibitors are potential candidates for anti-arthritis drugs. For the purposes of drug discovery, we reported the development and validation of fluorescence resonance energy transfer (FRET) assay for high-throughput screening (HTS) of the ADAMTS1 inhibitors...
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ژورنال
عنوان ژورنال: Journal of Bacteriology
سال: 2017
ISSN: 0021-9193,1098-5530
DOI: 10.1128/jb.00889-16